Begelomab (Biosimilar Reference Antibody) (DPP4)
Begelomab (Biosimilar Reference Antibody) (DPP4)

Catalog: 

RA0189

Target

DPP4/ADCP2/CD26

Isotype

IgG2b - kappa

Applications

ELISA;FC;Functional Assays;IF

Reactivities

Human

Size ($):

100 μg-50;1 mg-210;5 mg-500;10 mg-800;25 mg-1750;50 mg-3000;100 mg-4600

Data Sheet

Material Safety Data Sheet

Certificate of Analysis

Product Description

Begelomab is a murine (mouse) monoclonal antibody (typically IgG2b isotype) that specifically targets the Dipeptidyl Peptidase 4 (DPP4) receptor. It acts as an antagonist by binding to its target on the surface of T cells. This binding inhibits T-cell activation, proliferation, and most importantly, T-cell migration into tissues. Begelomab has been primarily investigated as an immunomodulatory agent for the treatment of severe, steroid-refractory acute Graft-versus-Host Disease (GvHD), a life-threatening complication following allogeneic hematopoietic stem cell transplantation (HSCT). By preventing the trafficking of pathogenic T cells, Begelomab aims to reduce GvHD-related tissue damage in the gut and skin.

Synonyms

BT 5/9, SAND 26, SAND-26, SAND26

CAS

1403744-56-8

Isotype

IgG2b - kappa

Host

Murine

Target

DPP4/ADCP2/CD26

Reactivity

Human

Expression System

CHO

Applications

ELISA, FC, Functional Assays, IF; Recommended dilution: FC, IF:1:200

Purity

>98% by SDS-PAGE

Concentration

Bottled at the concentration indicated on the vial.

Buffer

0.01M PBS, pH 7.4, contains no stabilizers or preservatives.

Endotoxin

<1.0 EU/mg as determined by LAL method

Conjugation

Non-conjugated

Formulation

Liquid or Lyophilized powder Note: We will preferentially ship the format that we have in stock, however, if you have any special requirement for the format, please remark your requirement when placing the order, we will prepare according to your demand.

Storage

store at -20°C or -80°C. Avoid repeated freeze.

Type

Antibody

Purposes

For research use only

References 1

Lorenzo RD, et, al. Begelomab for severe refractory dermatomyositis: A case report. Medicine (Baltimore). 2021 Mar 5;100(9):e24372.

References 2

Ojha R, et, al. Designing of a bispecific antibody against SARS-CoV-2 spike glycoprotein targeting human entry receptors DPP4 and ACE2. Hum Immunol. 2022 Apr;83(4):346-355.

References 3

References 4

References 5

Product Citations 1

Product Citations 2

https://pubmed.ncbi.nlm.nih.gov/33655912/
https://pubmed.ncbi.nlm.nih.gov/35042653/
https://www.oursmab.com/News/T-cell-activation-regulatory-factor-DPP4.html

Target Description

Synonyms

dipeptidyl-peptidase 4, dipeptidylpeptidase IV, adenosine deaminase complexing protein 2, ADCP2, TP103, T-cell activation antigen CD26, CD26

Biology Area

Immunology;CD Markers;Metabolism

Function

Dipeptidyl Peptidase 4 (DPP4/CD26), a multifunctional transmembrane glycoprotein with enzymatic, receptor, and co-stimulatory activities. It is constitutively expressed on the surface of various cell types, including T lymphocytes (particularly activated subsets), epithelial cells, and endothelial cells.

Additional Articles 1

T-cell-activation-regulatory-factor-DPP4

Additional Articles 2

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