Bentracimab (Biosimilar Reference Antibody) (Ticagrelor)
Bentracimab (Biosimilar Reference Antibody) (Ticagrelor)

Catalog: 

RA0728

Target

Ticagrelor

Isotype

Fab - G1 - lambda

Applications

Functional Assays

Reactivities

Drug

Size ($):

100 μg-50;1 mg-210;5 mg-500;10 mg-800;25 mg-1750;50 mg-3000;100 mg-4600

Data Sheet

Material Safety Data Sheet

Certificate of Analysis

Product Description

Bentracimab is an investigational, humanized monoclonal antibody fragment (Fab) designed as a specific reversal agent for the antiplatelet drug ticagrelor. It functions as a neutralizing antibody that binds with very high affinity to both ticagrelor and its active metabolite in the plasma, forming inactive complexes. This binding rapidly reverses the antiplatelet (P2Y12 receptor inhibitory) effects of ticagrelor, restoring platelet function. It is being developed for use in clinical scenarios where immediate reversal of ticagrelor's effects is required, such as in patients experiencing major bleeding or needing urgent surgery. It has demonstrated rapid and sustained reversal in Phase I and II trials.

Synonyms

MEDI2452, anti-ticagrelor, antidote for ticagrelor, MEDI-2452, PB-2452

CAS

2260568-31-6

Isotype

Fab - G1 - lambda

Host

Genetically human

Target

Ticagrelor

Reactivity

Drug

Expression System

CHO

Applications

Functional Assays;

Purity

>98% by SDS-PAGE

Concentration

Bottled at the concentration indicated on the vial.

Buffer

0.01M PBS, pH 7.4, contains no stabilizers or preservatives.

Endotoxin

<1.0 EU/mg as determined by LAL method

Conjugation

Non-conjugated

Formulation

Liquid or Lyophilized powder Note: We will preferentially ship the format that we have in stock, however, if you have any special requirement for the format, please remark your requirement when placing the order, we will prepare according to your demand.

Storage

store at -20°C or -80°C. Avoid repeated freeze.

Type

Antibody

Purposes

For research use only

References 1

Kathman SJ, et, al. Population pharmacokinetic-pharmacodynamic modeling of PB2452, a monoclonal antibody fragment being developed as a ticagrelor reversal agent, in healthy volunteers. CPT Pharmacometrics Syst Pharmacol. 2022 Jan;11(1):68-81.

References 2

Almquist J, et, al. Unraveling the pharmacokinetic interaction of ticagrelor and MEDI2452 (Ticagrelor antidote) by mathematical modeling. CPT Pharmacometrics Syst Pharmacol. 2016 Jun;5(6):313-23.

References 3

References 4

References 5

Product Citations 1

Product Citations 2

https://pubmed.ncbi.nlm.nih.gov/34713987/
https://pubmed.ncbi.nlm.nih.gov/27310493/

Target Description

Synonyms

BRILINTA® (US, Russia), BRILIQUE, POSSIA (EU)

Biology Area

Metabolism

Function

The target of Bentracimab is not an endogenous human protein or receptor, but the pharmacological drug ticagrelor (and its active metabolite). Ticagrelor is a direct-acting, reversible P2Y12 receptor antagonist used as an oral antiplatelet agent to prevent thrombotic events (e.g., in acute coronary syndrome).

Additional Articles 1

Additional Articles 2

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