Bifikafusp (Biosimilar Reference Antibody) (FN extracellular domain B)
Bifikafusp (Biosimilar Reference Antibody) (FN extracellular domain B)

Catalog: 

RA0255

Target

FN extracellular domain B

Isotype

scFv - heavy - kappa

Applications

ELISA;FC;Functional Assays;IF

Reactivities

Human

Size ($):

100 μg-50;1 mg-210;5 mg-500;10 mg-800;25 mg-1750;50 mg-3000;100 mg-4600

Data Sheet

Material Safety Data Sheet

Certificate of Analysis

Product Description

Bifikafusp alfa is an investigational immunocytokine, not a traditional monoclonal antibody. It is a fusion protein consisting of the human L19 antibody fragment (scFv) genetically fused to the cytokine human interleukin-2 (IL-2). The L19 fragment specifically targets the extra domain B (EDB) of fibronectin, a protein marker of tumor angiogenesis that is abundantly expressed in the neovasculature of most solid tumors but is virtually absent in normal adult tissues. The IL-2 component is a potent T-cell growth factor. This design allows for the targeted delivery of IL-2 directly to the tumor microenvironment, aiming to locally activate and expand tumor-infiltrating lymphocytes (TILs) and natural killer (NK) cells while minimizing the severe systemic toxicity associated with high-dose recombinant IL-2 therapy. It has demonstrated anticancer activity in clinical trials and is being evaluated for the treatment of various advanced solid tumors.

Synonyms

L19IL2, L19-IL-2, L19-IL2

CAS

1957239-90-5

Isotype

scFv - heavy - kappa

Host

Chimeric and/or humanised

Target

FN extracellular domain B

Reactivity

Human

Expression System

CHO

Applications

ELISA, FC, Functional Assays, IF; Recommended dilution: FC, IF:1:200

Purity

>98% by SDS-PAGE

Concentration

Bottled at the concentration indicated on the vial.

Buffer

0.01M PBS, pH 7.4, contains no stabilizers or preservatives.

Endotoxin

<1.0 EU/mg as determined by LAL method

Conjugation

Non-conjugated

Formulation

Liquid or Lyophilized powder Note: We will preferentially ship the format that we have in stock, however, if you have any special requirement for the format, please remark your requirement when placing the order, we will prepare according to your demand.

Storage

store at -20°C or -80°C. Avoid repeated freeze.

Type

Antibody

Purposes

For research use only

References 1

Wagner K, et, al. The targeted immunocytokine L19-IL2 efficiently inhibits the growth of orthotopic pancreatic cancer. Clin Cancer Res. 2008 Aug 1;14(15):4951-60.

References 2

References 3

References 4

References 5

Product Citations 1

Product Citations 2

https://pubmed.ncbi.nlm.nih.gov/18676770/

Target Description

Synonyms

FN (fibronectin) extra domain (EDB, ED-B)

Biology Area

Cancer Biology

Function

Fibronectin is a normal component of the extracellular matrix (ECM). The EDB domain is a splice variant that is highly and specifically expressed during embryonic development and in the neovasculature (newly formed blood vessels) of malignant tumors, but is undetectable in the ECM of healthy adult tissues (except for the endometrium and some placental structures). This makes EDB-fibronectin an excellent tumor angiogenesis marker. By utilizing the high-affinity L19 antibody fragment, bifikafusp alfa selectively homes to tumor blood vessels. Once localized, the fused IL-2 engages IL-2 receptors (primarily the high-affinity heterotrimeric receptor) on nearby immune cells, particularly CD8+ cytotoxic T cells and NK cells. This triggers their local activation, proliferation, and enhancement of cytotoxic function, creating a potent anti-tumor immune response directly within the tumor while sparing healthy tissues from systemic IL-2 exposure.

Additional Articles 1

Additional Articles 2

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