Cobolimab (Biosimilar Reference Antibody) (HAVCR2)
Cobolimab (Biosimilar Reference Antibody) (HAVCR2)
Cobolimab (Biosimilar Reference Antibody) (HAVCR2)-RA0281-Oursmab determined by SDS-PAGE. The purity of the protein is greater than 98%.
ELISA plate pre-coated Antigen protein, can bind Cobolimab (Biosimilar Reference Antibody) (HAVCR2)-RA0281 in a linear range of 3.91-125 ng/mL.
Cobolimab (Biosimilar Reference Antibody) (HAVCR2)

Catalog: 

RA0281

Target

HAVCR2/TIM3

Isotype

IgG4 - kappa

Applications

ELISA;FC;Functional Assays;IF

Reactivities

Human

Size ($):

100 μg-50;1 mg-210;5 mg-500;10 mg-800;25 mg-1750;50 mg-3000;100 mg-4600

Data Sheet

Material Safety Data Sheet

Certificate of Analysis

Product Description

Cobolimab is an investigational humanized IgG4 monoclonal antibody targeting the immune checkpoint receptor TIM-3 (T-cell immunoglobulin and mucin domain-containing protein 3). It is designed to enhance anti-tumor immunity by blocking this inhibitory pathway, which is often upregulated in exhausted T cells within the tumor microenvironment. With a potent mechanism of action that involves mediating the internalization of TIM-3 (with an IC₅₀ of 0.4464 nM), it represents a promising therapeutic strategy, particularly for solid tumors like non-small cell lung cancer (NSCLC), where it is being evaluated in clinical studies.

Synonyms

TSR-022

CAS

2022215-65-0

Isotype

IgG4 - kappa

Host

Humanised

Target

HAVCR2/TIM3

Reactivity

Human

Expression System

CHO

Applications

ELISA, FC, Functional Assays, IF; Recommended dilution: FC, IF:1:200

Purity

>98% by SDS-PAGE

Concentration

Bottled at the concentration indicated on the vial.

Buffer

0.01M PBS, pH 7.4, contains no stabilizers or preservatives.

Endotoxin

<1.0 EU/mg as determined by LAL method

Conjugation

Non-conjugated

Formulation

Liquid or Lyophilized powder Note: We will preferentially ship the format that we have in stock, however, if you have any special requirement for the format, please remark your requirement when placing the order, we will prepare according to your demand.

Storage

store at -20°C or -80°C. Avoid repeated freeze.

Type

Antibody

Purposes

For research use only

References 1

Falchook G S, et al. Phase 1 trial of TIM-3 inhibitor cobolimab monotherapy and in combination with PD-1 inhibitors nivolumab or dostarlimab (AMBER)[J]. 2022.

References 2

Markham A. Dostarlimab: First Approval. Drugs. 2021 Jul;81(10):1213-1219.

References 3

References 4

References 5

Product Citations 1

Product Citations 2

https://ascopubs.org/doi/abs/10.1200/JCO.2022.40.16_suppl.2504
https://pubmed.ncbi.nlm.nih.gov/34106455/
https://www.oursmab.com/News/T-cell-immunomodulatory-factor-TIM3.html

Target Description

Synonyms

hepatitis A virus cellular receptor 2, Tim-3, TIM3, FLJ14428, TIMD3, CD366

Biology Area

Immune Checkpoint;CD Markers;Immunology

Function

TIM-3, an immunoregulatory checkpoint receptor expressed on a subset of T cells (including exhausted and regulatory T cells), natural killer (NK) cells, monocytes, and dendritic cells. TIM-3 has multiple ligands, including galectin-9, CEACAM1, HMGB1, and phosphatidylserine. In the tumor microenvironment, the engagement of TIM-3 by its ligands (e.g., galectin-9 expressed by tumor or stromal cells) transmits an inhibitory signal that suppresses T-cell activation, cytokine production, and cytotoxic function, contributing to T-cell exhaustion and immune evasion.

Additional Articles 1

T-cell-immunomodulatory-factor-TIM3

Additional Articles 2

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