Glenzocimab (Biosimilar Reference Antibody) (GP6)
Glenzocimab (Biosimilar Reference Antibody) (GP6)

Catalog: 

RA0276

Target

GP6

Isotype

Fab - G1 - kappa

Applications

ELISA;FC;Functional Assays;IF

Reactivities

Human

Size ($):

100 μg-50;1 mg-210;5 mg-500;10 mg-800;25 mg-1750;50 mg-3000;100 mg-4600

Data Sheet

Material Safety Data Sheet

Certificate of Analysis

Product Description

Glenzocimab (development code ACT-017) is an investigational, humanized monoclonal antibody fragment (Fab) developed for the treatment of acute ischemic stroke and potentially other thrombotic conditions. It functions as a novel antiplatelet agent with a unique mechanism of action. Unlike traditional antiplatelet drugs that target platelet activation pathways (e.g., P2Y12 or COX-1 inhibition), glenzocimab is a selective inhibitor of platelet glycoprotein VI (GPVI). By binding to GPVI on the surface of platelets, it blocks the primary receptor for collagen, a key protein exposed at sites of vascular injury. This inhibition prevents collagen-induced platelet activation and thrombus formation without completely impairing hemostasis, aiming to reduce the risk of intracranial hemorrhage (bleeding), a major concern in stroke therapy.

Synonyms

ACT-017, ACT017

CAS

2101829-58-5

Isotype

Fab - G1 - kappa

Host

Humanised

Target

GP6

Reactivity

Human

Expression System

CHO

Applications

ELISA, FC, Functional Assays, IF; Recommended dilution: FC, IF:1:200

Purity

>98% by SDS-PAGE

Concentration

Bottled at the concentration indicated on the vial.

Buffer

0.01M PBS, pH 7.4, contains no stabilizers or preservatives.

Endotoxin

<1.0 EU/mg as determined by LAL method

Conjugation

Non-conjugated

Formulation

Liquid or Lyophilized powder Note: We will preferentially ship the format that we have in stock, however, if you have any special requirement for the format, please remark your requirement when placing the order, we will prepare according to your demand.

Storage

store at -20°C or -80°C. Avoid repeated freeze.

Type

Antibody

Purposes

For research use only

References 1

Wichaiyo S, et al. Glenzocimab: A GPVI (Glycoprotein VI)-Targeted Potential Antiplatelet Agent for the Treatment of Acute Ischemic Stroke. Stroke. 2022 Nov;53(11):3506-3513.

References 2

Lebozec K, et al. Design, development and characterization of ACT017, a humanized Fab that blocks platelet's glycoprotein VI function without causing bleeding risks. MAbs. 2017 Aug/Sep;9(6):945-958.

References 3

References 4

References 5

Product Citations 1

Product Citations 2

https://pubmed.ncbi.nlm.nih.gov/36128904/
https://pubmed.ncbi.nlm.nih.gov/28598281/
https://www.oursmab.com/News/The-platelet-glycoprotein-GP6.html

Target Description

Synonyms

glycoprotein VI platelet

Biology Area

Hematology;Immunology

Function

Glycoprotein VI (GPVI), a platelet-specific immunoglobulin (Ig) superfamily receptor that serves as the major signaling receptor for collagen. When the vascular endothelium is damaged (e.g., in an atherosclerotic plaque rupture leading to stroke), subendothelial collagen is exposed. Collagen binding to GPVI triggers a powerful intracellular signaling cascade via the Fc receptor gamma-chain (FcRγ), leading to platelet activation, shape change, granule release, and aggregation—forming a platelet-rich thrombus that can occlude cerebral arteries.

Additional Articles 1

The-platelet-glycoprotein-GP6

Additional Articles 2

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