Golocdacimab (Biosimilar Reference Antibody) (OLR1)
Golocdacimab (Biosimilar Reference Antibody) (OLR1)-RA0538-Oursmab determined by SDS-PAGE. The purity of the protein is greater than 98%.
Golocdacimab (Biosimilar Reference Antibody) (OLR1)

Catalog: 

RA0538

Target

OLR1/LOX1

Isotype

IgG1 - lambda

Applications

ELISA;FC;Functional Assays;IF

Reactivities

Human

Size ($):

100 μg-50;1 mg-210;5 mg-500;10 mg-800;25 mg-1750;50 mg-3000;100 mg-4600

Data Sheet

Material Safety Data Sheet

Certificate of Analysis

Product Description

Golocdacimab (development code MEDI6570) is an investigational, fully human monoclonal antibody being developed for the potential treatment of cardiometabolic diseases, specifically type 2 diabetes (T2D) and its associated complications. It functions as a targeted inhibitor of Lectin-like oxidized low-density lipoprotein receptor-1 (LOX-1). By binding with high affinity to LOX-1, golocdacimab blocks its interaction with its primary ligand, oxidized low-density lipoprotein (oxLDL). This blockade aims to inhibit the LOX-1-mediated signaling cascade that contributes to endothelial dysfunction, vascular inflammation, and atherogenesis—pathological processes that are accelerated in type 2 diabetes and drive cardiovascular risk.

Synonyms

MEDI-6570, MEDI 6570, MEDI6570

CAS

2418540-63-1

Isotype

IgG1 - lambda

Host

Genetically human

Target

OLR1/LOX1

Reactivity

Human

Expression System

CHO

Applications

ELISA, FC, Functional Assays, IF; Recommended dilution: FC, IF:1:200

Purity

>98% by SDS-PAGE

Concentration

Bottled at the concentration indicated on the vial.

Buffer

0.01M PBS, pH 7.4, contains no stabilizers or preservatives.

Endotoxin

<1.0 EU/mg as determined by LAL method

Conjugation

Non-conjugated

Formulation

Liquid or Lyophilized powder Note: We will preferentially ship the format that we have in stock, however, if you have any special requirement for the format, please remark your requirement when placing the order, we will prepare according to your demand.

Storage

store at -20°C or -80°C. Avoid repeated freeze.

Type

Antibody

Purposes

For research use only

References 1

Vavere AL, et al. Lectin-Like Oxidized Low-Density Lipoprotein Receptor 1 Inhibition in Type 2 Diabetes: Phase 1 Results. J Am Heart Assoc. 2023 Feb 7;12(3):e027540.

References 2

Varma V, et al. Identification of Response Biomarkers and Signaling Pathways Associated With the LOX-1 Blockade by MEDI6570 in Type 2 Diabetes[J]. Circulation, 2022, 146(Suppl_1): A11971-A11971.

References 3

References 4

References 5

Product Citations 1

Product Citations 2

https://pubmed.ncbi.nlm.nih.gov/36688371/
https://www.ahajournals.org/doi/abs/10.1161/circ.146.suppl_1.11971
https://www.oursmab.com/News/Oxidized-low-density-lipoprotein-receptor-OLR1.html

Target Description

Synonyms

oxidized low density lipoprotein receptor 1, LOX-1, SCARE1, CLEC8A

Biology Area

Immunology;Metabolism

Function

Lectin-like oxidized low-density lipoprotein receptor-1 (LOX-1), also known as oxidized low-density lipoprotein receptor 1 (OLR1). LOX-1 is a type II transmembrane glycoprotein belonging to the C-type lectin family. It is primarily expressed on vascular endothelial cells, but also on macrophages, vascular smooth muscle cells, and platelets. Under normal physiological conditions, LOX-1 expression is low. However, in the setting of metabolic stress like hyperglycemia and dyslipidemia in type 2 diabetes, LOX-1 expression is dramatically upregulated. Its main ligand, oxidized LDL (oxLDL), is a key component of diabetic dyslipidemia.

Additional Articles 1

Oxidized-low-density-lipoprotein-receptor-OLR1

Additional Articles 2

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